产品名称

英文名称：Tolterodine tartrate

同义词

Tolterodine tartrate、124937-52-6、Detrol LA、Detrol、Detrusitol、Tolterodine L-Tartrate、PNU-200583E、(R)-2-(3-(Diisopropylamino)-1-phenylpropyl)-4-methylphenol (2R,3R)-2,3-dihydroxysuccinate、UNII-5T619TQR3R、Tolterodine tartrate [USAN]、Tolterodine (tartrate)、Ka、酒石酸托特罗定

产品性质

CAS编号：124937-52-6

分子式：C22H31NO.C4H6O6

分子量：475.57

PubChem编号：443878

别名：酒石酸托特罗定

英文别名：Tolterodine tartrate|124937-52-6|Detrol LA|Detrol|Detrusitol|Tolterodine L-Tartrate|PNU-200583E|(R)-2-(3-(Diisopropylamino)-1-phenylpropyl)-4-methylphenol (2R,3R)-2,3-dihydroxysuccinate|UNII-5T619TQR3R|Tolterodine tartrate [USAN]|Tolterodine (tartrate)|Ka

规格或纯度：≥98%

英文名称：Tolterodine tartrate

生化机理：Tolterodine L-Tartrate is a muscarinic receptor antagonist that is active at all mAChR M subtypes. This compound blocks the opening of ion channels by acetylcholine, which in turn leads to muscle relaxation by blocking neuronal signaling. Tolterodine L-Tartrate is an inhibitor of mAChR M1, mAChR M2, mAChR M3, mAChR M4 and mAChR M5.

储存温度：2-8°C储存

运输条件：冰袋运输

备注：50mg、250mg、10mg、100mg卖完停产，不再备货

产品介绍：Tolterodine tartrate是Tolterodine的酒石酸盐形式，是一种竞争性的毒蕈碱型乙酰胆碱受体拮抗剂。A muscarinic receptor antagonist.Tolterodine tartrate is a tartrate salt of tolterodine that is a competitive muscarinic receptor antagonist.A muscarinic receptor antagonist.

IUPAC Name：(2R,3R)-2,3-dihydroxybutanedioic acid;2-[(1R)-3-[di(propan-2-yl)amino]-1-phenylpropyl]-4-methylphenol

INCHI：InChI=1S/C22H31NO.C4H6O6/c1-16(2)23(17(3)4)14-13-20(19-9-7-6-8-10-19)21-15-18(5)11-12-22(21)24;5-1(3(7)8)2(6)4(9)10/h6-12,15-17,20,24H,13-14H2,1-5H3;1-2,5-6H,(H,7,8)(H,9,10)/t20-;1-,2-/m11/s1

InChi Key：TWHNMSJGYKMTRB-KXYUELECSA-N

Canonical SMILES：CC1=CC(=C(C=C1)O)C(CCN(C(C)C)C(C)C)C2=CC=CC=C2.C(C(C(=O)O)O)(C(=O)O)O

Isomeric SMILES：CC1=CC(=C(C=C1)O)[C@H](CCN(C(C)C)C(C)C)C2=CC=CC=C2.[C@@H]([C@H](C(=O)O)O)(C(=O)O)O

PubChem CID：443878

溶解性：Soluble in water (0.012 mg/ml), DMSO (≥20 mg/ml), methanol, and ethanol (6 mg/ml)

象形图：

信号词：Danger

危险声明：H301 Toxic if swallowedH411 Toxic to aquatic life with long lasting effectsH302 Harmful if swallowedH361 Suspected of damaging fertility or the unborn child

预防措施声明：P273,P280,P321,P405,P501,P264,P270,P391,P330,P203,P301+P316,P301+P317,P318

产品包装